From Wikipedia, the free encyclopedia
| Names | |
|---|---|
| IUPAC name
1-(2-Cyclohexylphenoxy)-3-(propan-2-ylamino)propan-2-ol
| |
| Other names
Esprolol
| |
| Identifiers | |
3D model (JSmol)
|
|
| ChemSpider | |
| KEGG | |
PubChem CID
|
|
| UNII | |
CompTox Dashboard (EPA)
|
|
| |
| |
| Properties | |
| C18H29NO2 | |
| Molar mass | 291.435 g·mol−1 |
Except where otherwise noted, data are given for materials in their standard state (at 25 °C [77 °F], 100 kPa).
| |
Chemical compound
Exaprolol is a beta-adrenoceptor antagonist.[1]
Synthesis
[edit]
References
[edit]- ^ Van Waarde, A; Doorduin, J; De Jong, JR; Dierckx, RA; Elsinga, PH (2008). "Synthesis and preliminary evaluation of (S)-11C-exaprolol, a novel beta-adrenoceptor ligand for PET". Neurochemistry International. 52 (4–5): 729–33. doi:10.1016/j.neuint.2007.09.009. PMID 17961850.
- ^ Carissimi, M; Gentili, P; Grumelli, E; Milla, E; Picciola, G; Ravenna, F (1976). "Basic ethers of cyclohexylphenols with beta-blocking activity: Synthesis and pharmacological study of exaprolol". Arzneimittel-Forschung. 26 (4): 506–16. PMID 8056.
This drug article relating to the cardiovascular system is a stub. You can help Wikipedia by adding missing information. |
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