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  1. World Encyclopedia
  2. GABAergic - Wikipedia
GABAergic - Wikipedia
From Wikipedia, the free encyclopedia
Affecting GABA systems in the brain

In molecular biology and physiology, something is GABAergic or GABAnergic if it pertains to or affects the neurotransmitter gamma-aminobutyric acid (GABA). For example, a synapse is GABAergic if it uses GABA as its neurotransmitter, and a GABAergic neuron produces GABA. A substance is GABAergic if it produces its effects via interactions with the GABA system, such as by stimulating or blocking neurotransmission.

A GABAergic or GABAnergic agent is any chemical that modifies the effects of GABA in the body or brain. Some different classes of GABAergic drugs include agonists, antagonists, modulators, reuptake inhibitors and enzymes.[1]

See also

[edit]
  • Adenosinergic
  • Adrenergic
  • Cannabinoidergic
  • Cholinergic
  • Dopaminergic
  • Glutamatergic
  • Glycinergic
  • Histaminergic
  • Melatonergic
  • Monoaminergic
  • Neurotransmission
  • Opioidergic
  • Serotonergic

References

[edit]
  1. ^ Froestl, Wolfgang (2011). "An historical perspective on GABAergic drugs". Future Medicinal Chemistry. 3 (2): 163–175. doi:10.4155/fmc.10.285. ISSN 1756-8919. PMID 21428811.
  • v
  • t
  • e
GABA receptor modulators
Ionotropic
GABAATooltip γ-Aminobutyric acid A receptor
  • Agonists: 4-AHP
  • (+)-Catechin
  • Bamaluzole
  • Barbiturates (e.g., phenobarbital)
  • Beta-Alanine
  • BL-1020
  • DAVA
  • DH-P4S
  • Dihydromuscimol
  • GABA
  • Gabamide
  • GABOB
  • Gaboxadol (THIP)
  • Homotaurine (tramiprosate, 3-APS)
  • IAA (IMA)
  • Ibotenic acid
  • iso-THAZ
  • Isoguvacine
  • Isonipecotic acid
  • Kojic amine
  • L-838,417
  • Lignans (e.g., honokiol)
  • Methylglyoxal
  • Monastrol
  • Muscimol
  • Nefiracetam
  • Neuroactive steroids (e.g., allopregnanolone)
  • Org 20599
  • PF-6372865
  • Phenibut
  • Picamilon
  • 4-PIOL
  • P4S
  • Progabide
  • Propofol
  • Quisqualamine
  • SL-75102
  • Taurine
  • TACA
  • TAMP
  • Terpenoids (e.g., borneol)
  • Thio-4-PIOL
  • Thiomuscimol
  • Tolgabide
  • ZAPA
  • Positive modulators (abridged; see here for a full list): α-EMTBL
  • Alcohols (e.g., drinking alcohol, 2M2B)
  • Anabolic steroids
  • Avermectins (e.g., ivermectin)
  • Barbiturates (e.g., phenobarbital)
  • Benzodiazepines (e.g., diazepam)
  • Bromide compounds (e.g., potassium bromide)
  • Carbamates (e.g., meprobamate)
  • Carbamazepine
  • Chloralose
  • Chlormezanone
  • Clomethiazole
  • Dihydroergolines (e.g., ergoloid (dihydroergotoxine))
  • Etazepine
  • Etifoxine
  • Fenamates (e.g., mefenamic acid)
  • Flavonoids (e.g., apigenin, hispidulin)
  • Fluoxetine
  • Flupirtine
  • Imidazoles (e.g., etomidate)
  • Kava constituents (e.g., kavain)
  • Lanthanum
  • Loreclezole
  • Monastrol
  • Neuroactive steroids (e.g., allopregnanolone, cholesterol, THDOC)
  • Niacin
  • Niacinamide
  • Nonbenzodiazepines (e.g., β-carbolines (e.g., abecarnil), cyclopyrrolones (e.g., zopiclone), imidazopyridines (e.g., zolpidem), pyrazolopyrimidines (e.g., zaleplon))
  • Norfluoxetine
  • Petrichloral
  • Phenols (e.g., propofol)
  • Phenytoin
  • Piperidinediones (e.g., glutethimide)
  • Propanidid
  • Pyrazolopyridines (e.g., etazolate)
  • Quinazolinones (e.g., methaqualone)
  • Retigabine (ezogabine)
  • ROD-188
  • Skullcap constituents (e.g., baicalin)
  • Stiripentol
  • Sulfonylalkanes (e.g., sulfonmethane (sulfonal))
  • Topiramate
  • Valerian constituents (e.g., valerenic acid)
  • Volatiles/gases (e.g., chloral hydrate, chloroform, diethyl ether, paraldehyde, sevoflurane)
  • Antagonists: Bicuculline
  • Coriamyrtin
  • Dihydrosecurinine
  • Famiraprinium
  • Gabazine (SR-95531)
  • Hydrastine
  • Hyenanchin (mellitoxin)
  • Iso-THIP
  • PHP-501
  • Pitrazepin
  • Securinine
  • Sinomenine
  • SR-42641
  • THAZ
  • Thio-4-PIOL
  • Thio-THIP
  • Thiocolchicoside
  • Tutin
  • Negative modulators: 1,3M1B
  • 3M2B
  • 11-Ketoprogesterone
  • 17-Phenylandrostenol
  • α3IA
  • α5IA (LS-193,268)
  • β-CCB
  • β-CCE
  • β-CCM
  • β-CCP
  • β-EMGBL
  • Anabolic steroids
  • Amiloride
  • Anisatin
  • β-Lactams (e.g., penicillins, cephalosporins, carbapenems)
  • Basmisanil
  • Bemegride
  • Bicyclic phosphates (TBPS, TBPO, IPTBO)
  • BIDN
  • Bilobalide
  • Bupleurotoxin
  • Bupropion
  • CHEB
  • Chlorophenylsilatrane
  • Cicutoxin
  • Cloflubicyne
  • Cyclothiazide
  • DHEA
  • DHEA-S
  • Dieldrin
  • (+)-DMBB
  • DMCM
  • DMPC
  • EBOB
  • Etbicyphat
  • FG-7142 (ZK-31906)
  • Fiproles (e.g., fipronil)
  • Flavonoids (e.g., amentoflavone, oroxylin A)
  • Flumazenil
  • Fluoroquinolones (e.g., ciprofloxacin)
  • Flurothyl
  • Furosemide
  • Golexanolone
  • Iomazenil (123I)
  • IPTBO
  • Isopregnanolone (sepranolone)
  • L-655,708
  • Laudanosine
  • Lindane
  • MaxiPost
  • Morphine
  • Morphine-3-glucuronide
  • MRK-016
  • Naloxone
  • Naltrexone
  • Nicardipine
  • Nonsteroidal antiandrogens (e.g., apalutamide, bicalutamide, enzalutamide, flutamide, nilutamide)
  • Oenanthotoxin
  • Pentylenetetrazol (pentetrazol)
  • Phenylsilatrane
  • Picrotoxin (i.e., picrotin, picrotoxinin and dihydropicrotoxinin)
  • PNV-001
  • Pregnenolone sulfate
  • Propybicyphat
  • PWZ-029
  • Radequinil
  • Ro 15-4513
  • Ro 19-4603
  • RO4882224
  • RO4938581
  • Sarmazenil
  • SCS
  • Suritozole
  • TB-21007
  • TBOB
  • TBPS
  • TCS-1105
  • Terbequinil
  • TETS
  • Thujone
  • U-93631
  • Zinc
  • ZK-93426
GABAA-ρTooltip γ-Aminobutyric acid A-rho receptor
  • Agonists: BL-1020
  • CACA
  • CAMP
  • Homohypotaurine
  • GABA
  • GABOB
  • Ibotenic acid
  • Isoguvacine
  • Muscimol
  • N4-Chloroacetylcytosine arabinoside
  • Picamilon
  • Progabide
  • TACA
  • TAMP
  • Thiomuscimol
  • Tolgabide
  • Positive modulators: Allopregnanolone
  • Alphaxolone
  • ATHDOC
  • Lanthanides
  • Antagonists: (S)-2-MeGABA
  • (S)-4-ACPBPA
  • (S)-4-ACPCA
  • 2-MeTACA
  • 3-APMPA
  • 4-ACPAM
  • 4-GBA
  • cis-3-ACPBPA
  • Aza-THIP
  • CGP-36742 (SGS-742)
  • DAVA
  • Gabazine (SR-95531)
  • Gaboxadol (THIP)
  • I4AA
  • Iso-THIP
  • Isonipecotic acid
  • Loreclezole
  • P4MPA
  • P4S
  • SKF-97541
  • SR-95318
  • SR-95813
  • THAZ
  • Thio-THIP
  • TPMPA
  • trans-3-ACPBPA
  • ZAPA
  • Negative modulators: 5α-Dihydroprogesterone
  • Bilobalide
  • Loreclezole
  • Picrotoxin (picrotin, picrotoxinin)
  • Pregnanolone
  • ROD-188
  • THDOC
  • Zinc
Metabotropic
GABABTooltip γ-Aminobutyric acid B receptor
  • Agonists: 1,4-Butanediol
  • 3-APPA
  • 4-Fluorophenibut
  • Aceburic acid
  • Arbaclofen
  • Arbaclofen placarbil
  • Baclofen
  • BL-1020
  • GABA
  • Gabamide
  • GABOB
  • GBL
  • GHB
  • GHBAL
  • GHV
  • GVL
  • Isovaline
  • JZP-386
  • Lesogaberan
  • Phenibut
  • Picamilon
  • Progabide
  • Sodium oxybate
  • SKF-97,541
  • SL 75102
  • Tolgabide
  • Tolibut
  • Valiloxybate (XW-10172)
  • Positive modulators: ADX-71441
  • ASP-8062
  • BHF-177
  • BHFF
  • rac-BHFF
  • BSPP
  • CGP-7930
  • CGP-13501
  • GS-39783
  • INDV-1000
  • KK-92A
  • Antagonists: 2-Hydroxysaclofen
  • CGP-35348
  • CGP-36742
  • CGP-46381
  • CGP-52432
  • CGP-54626
  • CGP-55845
  • CGP-64213
  • DAVA
  • Homotaurine (tramiprosate, 3-APS)
  • Phaclofen
  • Saclofen
  • SCH-50911
  • Negative modulators: Compound 14
See also
Receptor/signaling modulators
GABAA receptor positive modulators
GABA metabolism/transport modulators
  • v
  • t
  • e
GABAA receptor positive modulators
Alcohols
  • Brometone
  • Butanol
  • Chloralodol
  • Chlorobutanol (cloretone)
  • Ethanol (alcohol) (alcoholic drink)
  • Ethchlorvynol
  • Isobutanol
  • Isopropanol
  • Menthol
  • Methanol
  • Methylpentynol
  • Pentanol
  • Petrichloral
  • Propanol
  • tert-Butanol (2M2P)
  • tert-Pentanol (2M2B)
  • Tribromoethanol
  • Trichloroethanol
  • Triclofos
  • Trifluoroethanol
Barbiturates
  • (-)-DMBB
  • Allobarbital
  • Alphenal
  • Amobarbital
  • Aprobarbital
  • Barbexaclone
  • Barbital
  • Benzobarbital
  • Benzylbutylbarbiturate
  • Brallobarbital
  • Brophebarbital
  • Butabarbital/Secbutabarbital
  • Butalbital
  • Buthalital
  • Butobarbital
  • Butallylonal
  • Carbubarb
  • Crotylbarbital
  • Cyclobarbital
  • Cyclopentobarbital
  • Difebarbamate
  • Enallylpropymal
  • Ethallobarbital
  • Eterobarb
  • Febarbamate
  • Heptabarb
  • Heptobarbital
  • Hexethal
  • Hexobarbital
  • Methallatal
  • Metharbital
  • Methitural
  • Methohexital
  • Methylphenobarbital
  • Narcobarbital
  • Nealbarbital
  • Pentobarbital
  • Phenallymal
  • Phenobarbital
  • Phetharbital
  • Primidone
  • Probarbital
  • Propallylonal
  • Propylbarbital
  • Proxibarbital
  • Reposal
  • Secobarbital
  • Sigmodal
  • Spirobarbital
  • Talbutal
  • Tetrabamate
  • Tetrabarbital
  • Thialbarbital
  • Thiamylal
  • Thiobarbital
  • Thiobutabarbital
  • Thiopental
  • Thiotetrabarbital
  • Valofane
  • Vinbarbital
  • Vinylbital
Benzodiazepines
  • 2-Oxoquazepam
  • 3-Hydroxyphenazepam
  • Adinazolam
  • Alprazolam
  • Arfendazam
  • Avizafone
  • Bentazepam
  • Bretazenil
  • Bromazepam
  • Bromazolam
  • Brotizolam
  • Camazepam
  • Carburazepam
  • Chlordiazepoxide
  • Ciclotizolam
  • Cinazepam
  • Cinolazepam
  • Clazolam
  • Climazolam
  • Clobazam
  • Clonazepam
  • Clonazolam
  • Cloniprazepam
  • Clorazepate
  • Clotiazepam
  • Cloxazolam
  • CP-1414S
  • Cyprazepam
  • Delorazepam
  • Demoxepam
  • Diazepam
  • Diclazepam
  • Dimdazenil
  • Doxefazepam
  • Elfazepam
  • Estazolam
  • Ethyl carfluzepate
  • Ethyl dirazepate
  • Ethyl loflazepate
  • Etizolam
  • FG-8205
  • Fletazepam
  • Flubromazepam
  • Flubromazolam
  • Fludiazepam
  • Flunitrazepam
  • Flunitrazolam
  • Flurazepam
  • Flutazolam
  • Flutemazepam
  • Flutoprazepam
  • Fosazepam
  • Gidazepam
  • Halazepam
  • Haloxazolam
  • Iclazepam
  • Imidazenil
  • Irazepine
  • Ketazolam
  • Lofendazam
  • Lopirazepam
  • Loprazolam
  • Lorazepam
  • Lormetazepam
  • Meclonazepam
  • Medazepam
  • Menitrazepam
  • Metaclazepam
  • Mexazolam
  • Midazolam
  • Motrazepam
  • N-Desalkylflurazepam
  • Nifoxipam
  • Nimetazepam
  • Nitrazepam
  • Nitrazepate
  • Nitrazolam
  • Nordazepam
  • Nortetrazepam
  • Oxazepam
  • Oxazolam
  • Phenazepam
  • Pinazepam
  • Pivoxazepam
  • Prazepam
  • Premazepam
  • Proflazepam
  • Pyrazolam
  • QH-II-66
  • Quazepam
  • Reclazepam
  • Remimazolam
  • Rilmazafone
  • Ripazepam
  • Ro48-6791
  • Ro48-8684
  • SH-053-R-CH3-2′F
  • Sulazepam
  • Temazepam
  • Tetrazepam
  • Tolufazepam
  • Triazolam
  • Triflubazam
  • Triflunordazepam (Ro5-2904)
  • Tuclazepam
  • Uldazepam
  • Zapizolam
  • Zolazepam
  • Zomebazam
Carbamates
  • Carisbamate
  • Carisoprodol
  • Clocental
  • Cyclarbamate
  • Difebarbamate
  • Emylcamate
  • Ethinamate
  • Febarbamate
  • Felbamate
  • Hexapropymate
  • Hydroxyphenamate
  • Lorbamate
  • Mebutamate
  • Meprobamate
  • Nisobamate
  • Pentabamate
  • Phenprobamate
  • Procymate
  • Styramate
  • Tetrabamate
  • Tybamate
Flavonoids
  • 6-Methylapigenin
  • Ampelopsin (dihydromyricetin)
  • Apigenin
  • Baicalein
  • Baicalin
  • Catechin
  • EGC
  • EGCG
  • Hispidulin
  • Linarin
  • Luteolin
  • Rc-OMe
  • Skullcap constituents (e.g., baicalin)
  • Wogonin
Imidazoles
  • Etomidate
  • Metomidate
  • Methoxyetomidate
  • Propoxate
  • Isopropoxate
  • Butomidate
  • Iso-butomidate
  • Sec-butomidate
  • CF2-Etomidate
  • CF3-Etomidate
  • CF3-Propoxate
  • Flutomidate
  • 2,6-Dichloro-3-fluoroetomidate
Kava constituents
  • 10-Methoxyyangonin
  • 11-Methoxyyangonin
  • 11-Hydroxyyangonin
  • Desmethoxyyangonin
  • 11-Methoxy-12-hydroxydehydrokavain
  • 7,8-Dihydroyangonin
  • Kavain
  • 5-Hydroxykavain
  • 5,6-Dihydroyangonin
  • 7,8-Dihydrokavain
  • 5,6,7,8-Tetrahydroyangonin
  • 5,6-Dehydromethysticin
  • Methysticin
  • 7,8-Dihydromethysticin
  • Yangonin
Monoureides
  • Acecarbromal
  • Apronal (apronalide)
  • Bromisoval
  • Carbromal
  • Capuride
  • Ectylurea
Neuroactive steroids
  • Acebrochol
  • Allopregnanolone (brexanolone)
  • Alfadolone
  • Alfaxalone
  • 3α-Androstanediol
  • Androstenol
  • Androsterone
  • Certain anabolic-androgenic steroids
  • Cholesterol
  • DHDOC
  • 3α-DHP
  • 5α-DHP
  • 5β-DHP
  • DHT
  • Etiocholanolone
  • Ganaxolone
  • Hydroxydione
  • Minaxolone
  • ORG-20599
  • ORG-21465
  • P1-185
  • Posovolone
  • Pregnanolone (eltanolone)
  • Progesterone
  • Renanolone
  • SAGE-105
  • SAGE-324
  • SAGE-516
  • SAGE-689
  • SAGE-872
  • Testosterone
  • THDOC
  • Zuranolone
Nonbenzodiazepines
  • Cyclopyrrolones: Eszopiclone
  • Pagoclone
  • Pazinaclone
  • Suproclone
  • Suriclone
  • Zopiclone
  • Imidazopyridines: Alpidem
  • DS-1
  • Necopidem
  • Saripidem
  • Zolpidem
  • Pyrazolopyrimidines: Divaplon
  • Fasiplon
  • Indiplon
  • Lorediplon
  • Ocinaplon
  • Panadiplon
  • Taniplon
  • Zaleplon
  • Others: Adipiplon
  • AXS-17 (BAER-101, AZD-7325)
  • CGS-8216
  • CGS-9896
  • CGS-13767
  • CGS-20625
  • CL-218,872
  • CP-615,003
  • CTP-354
  • ELB-139
  • GBLD-345
  • Imepitoin
  • JM-1232
  • L-838,417
  • Lirequinil (Ro41-3696)
  • Miltirone (rosmariquinone)
  • NS-2664
  • NS-2710
  • NS-11394
  • Pipequaline
  • ROD-188
  • RWJ-51204
  • SB-205,384
  • SX-3228
  • TGSC01AA
  • TP-003
  • TPA-023
  • TP-13
  • U-89843A
  • U-90042
  • Viqualine
  • Y-23684
Phenols
  • Cipepofol
  • Fospropofol
  • Propofol
  • Propofol hemisuccinate
  • Thymol
Piperidinediones
  • Glutethimide
  • Methyprylon
  • Piperidione
  • Pyrithyldione
Pyrazolopyridines
  • Cartazolate
  • Etazolate
  • ICI-190,622
  • Tracazolate
Quinazolinones
  • Afloqualone
  • Cloroqualone
  • Diproqualone
  • Etaqualone
  • Mebroqualone
  • Mecloqualone
  • Methaqualone
  • Methylmethaqualone
  • Nitromethaqualone
  • SL-164
Volatiles/gases
  • Acetone
  • Acetophenone
  • Acetylglycinamide chloral hydrate
  • Aliflurane
  • Benzene
  • Butane
  • Butylene
  • Centalun
  • Chloral
  • Chloral betaine
  • Chloral hydrate
  • Chloroform
  • Cryofluorane
  • Desflurane
  • Dichloralphenazone
  • Dichloromethane
  • Diethyl ether
  • Enflurane
  • Ethyl chloride
  • Ethylene
  • Fluroxene
  • Gasoline
  • Halopropane
  • Halothane
  • Isoflurane
  • Kerosine
  • Methoxyflurane
  • Methoxypropane
  • Nitric oxide
  • Nitrogen
  • Nitrous oxide
  • Norflurane
  • Paraldehyde
  • Propane
  • Propylene
  • Roflurane
  • Sevoflurane
  • Synthane
  • Teflurane
  • Toluene
  • Trichloroethane (methyl chloroform)
  • Trichloroethylene
  • Vinyl ether
Others/unsorted
  • 3-Hydroxybutanal
  • α-EMTBL
  • AA-29504
  • Alogabat
  • Avermectins (e.g., ivermectin)
  • Bromide compounds (e.g., lithium bromide, potassium bromide, sodium bromide)
  • Carbamazepine
  • Chloralose
  • Chlormezanone
  • Clomethiazole
  • Darigabat
  • DEABL
  • Deuterated etifoxine
  • Dihydroergolines (e.g., dihydroergocryptine, dihydroergosine, dihydroergotamine, ergoloid (dihydroergotoxine))
  • DS2
  • Efavirenz
  • Etazepine
  • Etifoxine
  • Fenamates (e.g., flufenamic acid, mefenamic acid, niflumic acid, tolfenamic acid)
  • Fluoxetine
  • Flupirtine
  • Hopantenic acid
  • KRM-II-81
  • Lanthanum
  • Lavender oil
  • Lignans (e.g., 4-O-methylhonokiol, honokiol, magnolol, obovatol)
  • Loreclezole
  • Menthyl isovalerate (validolum)
  • Monastrol
  • Nicotinic acid
  • Nicotinamide
  • Org 25,435
  • Phenytoin
  • Propanidid
  • Retigabine (ezogabine)
  • Safranal
  • Seproxetine
  • Stiripentol
  • Sulfonylalkanes (e.g., sulfonmethane (sulfonal), tetronal, trional)
  • Terpenoids (e.g., borneol)
  • Topiramate
  • Valerian constituents (e.g., isovaleric acid, isovaleramide, valerenic acid, valerenol)
  • Unsorted benzodiazepine site positive modulators: α-Pinene
  • MRK-409 (MK-0343)
  • TCS-1105
  • TCS-1205
See also: Receptor/signaling modulators • GABA receptor modulators • GABA metabolism/transport modulators
  • v
  • t
  • e
GABATooltip γ-Aminobutyric acid metabolism and transport modulators
Transporter
GATTooltip GABA transporter
  • Inhibitors: 4-Aminovaleric acid
  • β-Alanine
  • Arecaidine
  • CI-966
  • DABA
  • Deramciclane (EGIS-3886, EGYT-3886)
  • Dihydromuscimol
  • EF-1502
  • Gabaculine
  • Guvacine
  • Ibotenic acid
  • Muscimol
  • Nipecotic acid
  • NNC 05-2090
  • NO-711
  • Riluzole
  • SKF-89976A
  • SNAP-5114
  • TACA
  • THAO
  • Thio-THIP
  • Thio-THPO
  • THPO
  • Tiagabine
VIAATTooltip Vesicular inhibitory amino acid transporter
  • Inhibitors: β-Alanine
  • Bafilomycin A1
  • Chicago sky blue 6B
  • Evans blue
  • GABA
  • Glycine
  • N-Butyric acid
  • Nigericin
  • Nipecotic acid
  • Valinomycin
  • Vigabatrin
Enzyme
GADTooltip Glutamate decarboxylase
  • Inhibitors: 3-Mercaptopropionic acid
  • AAOA
  • L-Allylglycine
  • Semicarbazide
  • Activators: 3-Methyl-GABA
GABA-TTooltip γ-Aminobutyrate aminotransferase
  • Inhibitors: 3-Hydrazinopropionic acid
  • DABA
  • γ-Acetylenic-GABA
  • AOAA
  • EOS
  • Gabaculine
  • Isoniazid
  • L-Cycloserine
  • Phenelzine
  • PEH
  • Rosmarinic acid (lemon balm)
  • Sodium valproate
  • Valnoctamide
  • Valproate pivoxil
  • Valproate semisodium (divalproex sodium)
  • Valproic acid
  • Valpromide
  • Vigabatrin
  • Activators: 3-Methyl-GABA
Other
Antivitamin B6
  • Ginkgotoxin
See also
Receptor/signaling modulators
GABA receptor modulators
GABAA receptor positive modulators
Glutamate metabolism/transport modulators
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Pharmacomodulation
Types
  • ♦ Enzyme: Inducer
  • Inhibitor
  • ♦ Ion channel: Opener
  • Blocker
  • ♦ Receptor: Agonist
  • Partial agonist
  • Antagonist
  • Inverse agonist
  • Positive allosteric modulator (PAM)
  • Negative allosteric modulator (NAM)
  • ♦ Transporter [Reuptake vs Efflux]: Enhancer (RE)
  • Inhibitor (RI)
  • Releaser (RA)
  • ♦ Miscellaneous: Precursor
  • Cofactor
Classes
Enzyme
see Enzyme inhibition
Ion channel
See Ion channel modulators
Receptor &
transporter
BA/M
Adrenergic
  • Adrenergic receptor agonist (α
  • β (1
  • 2))
  • Adrenergic receptor antagonist (α (1
  • 2)
  • β)
  • Norepinephrine reuptake inhibitor (NRI)
Dopaminergic
  • Dopamine receptor agonist
  • Dopamine receptor antagonist
  • Dopamine reuptake inhibitor (DRI)
Histaminergic
  • Histamine receptor agonist
  • Histamine receptor antagonist (H1
  • H2
  • H3)
Serotonergic
  • Serotonin receptor agonist
  • Serotonin receptor antagonist (5-HT3)
  • Serotonin reuptake inhibitor (SRI)
AA
GABAergic
  • GABA receptor agonist
  • GABA receptor antagonist
  • GABA reuptake inhibitor (GRI)
Glutamatergic
  • Glutamate receptor agonist (AMPA)
  • Glutamate receptor antagonist (NMDA)
  • Glutamate reuptake inhibitor
Cholinergic
  • Acetylcholine receptor agonist (Muscarinic
  • Nicotinic)
    • Cholinesterase inhibitor
  • Acetylcholine receptor antagonist (Muscarinic
  • Nicotinic (Ganglionic
  • Muscular))
Cannabinoidergic
  • Cannabinoid receptor agonist
  • Cannabinoid receptor antagonist
  • Endocannabinoid enhancer (eCBE)
  • Endocannabinoid reuptake inhibitor (eCBRI)
Opioidergic
  • Opioid modulator
  • Opioid receptor agonist
  • Opioid receptor antagonist
  • Enkephalinase inhibitor
Other
  • Adenosine reuptake inhibitor (AdoRI)
  • Angiotensin II receptor antagonist
  • Endothelin receptor antagonist
  • NK1 receptor antagonist
  • Vasopressin receptor antagonist
Miscellaneous
  • Cofactor (see Enzyme cofactors)
  • Precursor (see Amino acids)


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This drug article relating to the nervous system is a stub. You can help Wikipedia by adding missing information.

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Categories:
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  • Neurotransmitters
  • Nervous system drug stubs
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Sunting pranala
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url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url url 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